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\u5168\u822c\u7684 Freiname \u30c1\u30b6\u30cb\u30b8\u30f3 \u4ed6\u306e\u540d\u524d 4-\u30af\u30ed\u30fc\u30eb – n – \uff084,5-dihydro-1 h -IMIDAZOL-2-ILL\uff09-8-THIA-7,9-\u30b8\u30a2\u30b6\u30d3\u30b7\u30af\u30ed[4.3.0]\u30ce\u30f3A-2,4,6,9-\u30c6\u30c8\u30e9\u30a8\u30f3-5-\u30a2\u30df\u30f3 \u30de\u30c3\u30b7\u30e5\u30d5\u30a9\u30fc\u30df\u30e5\u30e9 c 9 h 8 cln 5 s \uff08\u30c1\u30b6\u30cb\u30b8\u30f3\uff09 c 9 h 8 cln 5 S\u30fbHCl \uff08\u30c1\u30b6\u30cb\u30b8\u30f3\u30fb\u5869\u9178\u5869\uff09 \u5916\u90e8\u8b58\u5225\u5b50\/\u30c7\u30fc\u30bf\u30d9\u30fc\u30b9 \u85ac ATC\u30b3\u30fc\u30c9 M03 BX02 \u30a2\u30af\u30c6\u30a3\u30d6\u306a\u6210\u5206\u30af\u30e9\u30b9 \u7b4b\u8089\u306e\u518dx \u6a5f\u69cb a 2 – \u30a2\u30c9\u30ec\u30ce\u30bc\u30d7\u30bf\u30fc\u30a2\u30b4\u30cb\u30b9\u30c8 \u7279\u6027 \u30e2\u30eb\u8cea\u91cf 253.71 g\u30fbmol -1 \u7dcf\u72b6\u614b \u796d\u308a \u878d\u70b9 221\u2013223\u00b0C [\u521d\u3081] \u6eb6\u89e3\u5ea6 > 20 mg\/ml\u306e\u6c34 [2] 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\uff09\u3002 \u2191 Sirdalud\u00ae\u30b9\u30da\u30b7\u30e3\u30ea\u30b9\u30c8\u60c5\u5831\u3001Red List 2008\u3002 \u2191 rote-hand-brief Zu Sirdalud \uff08 \u8a18\u5ff5 2007\u5e7410\u670822\u65e5\u304b\u3089 \u30a4\u30f3\u30bf\u30fc\u30cd\u30c3\u30c8\u30a2\u30fc\u30ab\u30a4\u30d6 \uff09\u3002 \u2191 Granfors MT\u3001Backman JT\u3001Laitila J\u3001Neuvonen PJ\u3002 \u30a8\u30c1\u30cb\u30eb\u30a8\u30b9\u30c8\u30e9\u30b8\u30aa\u30fc\u30eb\u3068\u30b2\u30b9\u30c8\u30c7\u30f3\u3092\u542b\u3080\u7d4c\u53e3\u907f\u598a\u85ac\u306f\u3001\u30b7\u30c8\u30af\u30ed\u30e0P450 1A2\u3092\u963b\u5bb3\u3059\u308b\u3053\u3068\u306b\u3088\u308a\u3001\u8840\u6f3f\u6fc3\u5ea6\u3068\u30c1\u30b6\u30cb\u30b8\u30f3\u306e\u52b9\u679c\u3092\u8457\u3057\u304f\u5897\u52a0\u3055\u305b\u307e\u3059\u3002 Clin Pharmacol Ther\u3002 2005\u5e7410\u6708; 78\uff084\uff09\uff1a400-11\u3001 PMID 16198659 \u3002 \u2191 \u30c1\u30b6\u30cb\u30b8\u30f3\u5869\u9178\u30ab\u30d7\u30bb\u30eb\u3002 \u306e\uff1a dailymed\u3002 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